Sage Journals: Discover world-class research

Free access

Review article

First published 2020-2

High-Throughput Cellular Thermal Shift Assays in Research and Drug Discovery

Mark J. Henderson, Marc A. Holbert, Anton Simeonov [...]

Journal of Biomolecular Screening

Free access

Research article

First published 2020-2

Drug Target Engagement Using Coupled Cellular Thermal Shift Assay—Acoustic Reverse-Phase Protein Array

Adrien Herledan, Marine Andres, Aurore Lejeune-Dodge [...]

Journal of Biomolecular Screening

Free access

Research article

First published 2018-1

A High-Throughput Dose-Response Cellular Thermal Shift Assay for Rapid Screening of Drug Target Engagement in Living Cells,Exemplified Using SMYD3 and IDO1

Dean E. McNulty, William G. Bonnette, Hongwei Qi [...]

Journal of Biomolecular Screening

Free access

Research article

First published 2020-2

Perspective on CETSA Literature: Toward More Quantitative Data Interpretation

Brinton Seashore-Ludlow, Hanna Axelsson, Thomas Lundbäck

Journal of Biomolecular Screening

Open access

Research article

First published 2021-4

A Tale of Two Tails: Efficient Profiling of Protein Degraders by Specific Functional and Target Engagement Readouts

Alexey L. Chernobrovkin, Cindy Cázares-Körner, Tomas Friman [...]

Journal of Biomolecular Screening

Open access

Research article

First published 2019-2

Positioning High-Throughput CETSA in Early Drug Discovery through Screening against B-Raf and PARP1

Joseph Shaw, Ian Dale, Paul Hemsley [...]

Journal of Biomolecular Screening

Retricted access

Research article

First published 2021-12

A Genome-Edited ERα-HiBiT Fusion Reporter Cell Line for the Identification of ERα Modulators Via High-Throughput Screening and CETSA

Hunter G. Larson, Alexey V. Zakharov, Sukumar Sarkar [...]

ASSAY and Drug Development Technologies

Free access

Research article

First published 2016-12

Early Perspective

Brinton Seashore-Ludlow, Thomas Lundbäck

Journal of Biomolecular Screening

Free access

Research article

First published 2018-2

Cell Density Affects the Detection of Chk1 Target Engagement by the Selective Inhibitor V158411

Clara C. Geneste, Andrew J. Massey

Journal of Biomolecular Screening

Free access

Research article

First published 2015-2

Cell-Based Protein Stabilization Assays for the Detection of Interactions between Small-Molecule Inhibitors and BRD4

Jessica Schulze, Dieter Moosmayer, Joerg Weiske [...]

Journal of Biomolecular Screening

Search results