Sage Journals: Discover world-class research

Free access

Review article

First published 2015-6

Inhibition of bromodomain and extra-terminal proteins (BET) as a potential therapeutic approach in haematological malignancies: emerging preclinical and clinical evidence

Aristeidis Chaidos, Valentina Caputo, Anastasios Karadimitris

Therapeutic Advances in Hematology

Open access

Announcement

First published 2013

Stimulation of Hepatic Apolipoprotein A-I Production by Novel Thieno-Triazolodiazepines: Roles of the Classical Benzodiazepine Receptor,PAF Receptor,and Bromodomain Binding

Herman J. Kempen, Daniel Bellus, Oleg Fedorov [...]

Lipid Insights

Open access

Article commentary

First published 2020-11

Free as a BRD4: Bromodomain Inhibition Ameliorates Disease Phenotypes in a Model of MECP2 Deficiency and Is a Potential Therapy for Rett Syndrome

Kay-Marie Joan Lamar, Gemma L. Carvill

Epilepsy Currents

Retricted access

Research article

First published 2022-04

The BET Protein Inhibitor Apabetalone Rescues Diabetes-Induced Impairment of Angiogenic Response by Epigenetic Regulation of Thrombospondin-1

Shafeeq A. Mohammed, Mattia Albiero, Samuele Ambrosini [...]

Antioxidants & Redox Signaling

Free access

Research article

First published 2020-4

Preclinical Safety Assessment of a Highly Selective and Potent Dual Small-Molecule Inhibitor of CBP/P300 in Rats and Dogs

Paula Katavolos, Gary Cain, Cindy Farman [...]

Toxicologic Pathology

Free access

Research article

First published 2015-2

Cell-Based Protein Stabilization Assays for the Detection of Interactions between Small-Molecule Inhibitors and BRD4

Jessica Schulze, Dieter Moosmayer, Joerg Weiske [...]

Journal of Biomolecular Screening

Open access

Review article

First published 2014

Use of Epigenetic Drugs in Disease: An Overview

Sarah Heerboth, Karolina Lapinska, Nicole Snyder [...]

Epigenetics Insights

Free access

Research article

First published 2018-3

Cochlearoids L and M: Two New Meroterpenoids from the Fungus Ganoderma cochlear

Fu-Ying Qin, Yong-Ming Yan, Zheng-Chao Tu [...]

Natural Product Communications

Free access

Research article

First published 2021-5

Suppression of bromodomain-containing protein 4 protects trophoblast cells from oxidative stress injury by enhancing Nrf2 activation

Yiqing Wu, Yang Mi, Fan Zhang [...]

Human & Experimental Toxicology

Free access

Research article

First published 2015-3

BRD4 promotes tumor growth and epithelial-mesenchymal transition in hepatocellular carcinoma

Pengfei Zhang, Zhaoru Dong, Jiabin Cai [...]

International Journal of Immunopathology and Pharmacology

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