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Research article

First published 2017-8

Discovery of Novel Gq-Biased LPA1 Negative Allosteric Modulators

Yuji Shimizu, Masaharu Nakayama

Journal of Biomolecular Screening

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Research article

First published 2021-11-23

Positive and Negative Selective Allosteric Modulators of α5 GABA A Receptors: Effects on Emotionality,Motivation,and Motor Function in the 5xFAD Model of Alzheimer’s Disease

Jovana Aranđelović, Anja Santrač, Bojan Batinić [...]

Journal of Alzheimer’s Disease

Open access

Research article

First published 2024

Negative effect of treatment with mGluR5 negative allosteric modulator AFQ056 on blood biomarkers in young individuals with Fragile X syndrome

Dragana Protic, Elizabeth Breeze, Guadalupe Mendoza [...]

Sage Open Medicine

Free access

Research article

First published 2015-10

Drug-induced Skin Lesions in Cynomolgus Macaques Treated with Metabotropic Glutamate Receptor 5 (mGluR5) Negative Allosteric Modulators

Gopinath S. Palanisamy, John M. Marcek, Gregg D. Cappon [...]

Toxicologic Pathology

Open access

Research article

First published 2013-1

Effects of a Metabotropic Glutamate Receptor Subtype 7 Negative Allosteric Modulator in the Periaqueductal Grey on Pain Responses and Rostral Ventromedial Medulla Cell Activity in Rat

Enza Palazzo, Ida Marabese, Livio Luongo [...]

Molecular Pain

Retricted access

Review article

First published 2015-2

Dementia praecox redux: A systematic review of the nicotinic receptor as a target for cognitive symptoms of schizophrenia

Arann R Rowe, Louise Mercer, Valentina Casetti [...]

Journal of Psychopharmacology

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Research article

First published 2012-10

Development of a High-Throughput Calcium Flux Assay for Identification of All Ligand Types Including Positive,Negative,and Silent Allosteric Modulators for G Protein-Coupled Receptors

Devin J. Noblin, Robert L. Bertekap, Neil T. Burford [...]

ASSAY and Drug Development Technologies

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Review article

First published 2016-01

Allosteric Modulators of the CB 1 Cannabinoid Receptor: A Structural Update Review

Paula Morales, Pilar Goya, Nadine Jagerovic [...]

Cannabis & Cannabinoid Research

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Research article

First published 2016-08

Exploring the Benzimidazole Ring as a Substitution for Indole in Cannabinoid Allosteric Modulators

Laura Hernandez-Folgado, Lesley A. Stevenson, Paula Morales [...]

Cannabis & Cannabinoid Research

Free access

Research article

First published 2010-2

Development of a β-Lactamase Reporter Gene Assay for Metabotropic Glutamate Receptor 1 by Using Coexpression of Glutamate Transporter

Gentaroh Suzuki, Hiroshi Kawamoto, Hisashi Ohta

Journal of Biomolecular Screening

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