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Research article

First published 2025-6

A Characterization of the Nonclinical Pharmacology and Toxicology of Aficamten,a Reversible Allosteric Inhibitor of Cardiac Myosin

Michael K. Pugsley, Darren T. Hwee, Brett R. Winters [...]

International Journal of Toxicology

Free access

Research article

First published 2012-7

Detection of Allosteric Kinase Inhibitors by Displacement of Active Site Probes

Connie S. Lebakken, Laurie J. Reichling, Jason M. Ellefson [...]

Journal of Biomolecular Screening

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Research article

First published 2012-6

Development of an AlphaScreen-Based HIV-1 Integrase Dimerization Assay for Discovery of Novel Allosteric Inhibitors

Jonas Demeulemeester, Cristina Tintori, Maurizio Botta [...]

Journal of Biomolecular Screening

Open access

Research article

First published 2025

Phenazine Scaffolds as a Potential Allosteric Inhibitor of LasR Protein in Pseudomonas aeruginosa

Prisca Baah Nketia, Prince Manu, Priscilla Osei-Poku [...]

Bioinformatics and Biology Insights

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Research article

First published 2023-08

Positive Allosteric Modulation of Antithrombin's Inhibitory Activity by RNA Aptamers

Khalequz Zaman, Adi Breitman, Isa Malik [...]

Nucleic Acid Therapeutics

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Research article

First published 2021-03

Honokiol Bis-Dichloroacetate Is a Selective Allosteric Inhibitor of the Mitochondrial Chaperone TRAP1

Carlos Sanchez-Martin, Daniela Menon, Elisabetta Moroni [...]

Antioxidants & Redox Signaling

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Research article

First published 2015-12

High-Throughput Screening Strategy Identifies Allosteric,Covalent Human D-Amino Acid Oxidase Inhibitor

Ryan T. Terry-Lorenzo, Keiki Masuda, Kohtaroh Sugao [...]

Journal of Biomolecular Screening

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Research article

First published 2011-02

Virtual Ligand Screening of the National Cancer Institute (NCI) Compound Library Leads to the Allosteric Inhibitory Scaffolds of the West Nile Virus NS3 Proteinase

Sergey A. Shiryaev, Anton V. Cheltsov, Katarzyna Gawlik [...]

ASSAY and Drug Development Technologies

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Research article

First published

sAβPP α is a Potent Endogenous Inhibitor of BACE1

Clare Peters-Libeu, Jesus Campagna, Michael Mitsumori [...]

Journal of Alzheimer’s Disease

Open access

Research article

First published 2021

Ligand Docking Methods to Recognize Allosteric Inhibitors for G-Protein-Coupled Receptors

K Harini, S Jayashree, Vikas Tiwari [...]

Bioinformatics and Biology Insights

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