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Research article

First published 2019-11

Cortical 5-hydroxytryptamine 1A receptor biased agonist,NLX-101,displays rapid-acting antidepressant-like properties in the rat chronic mild stress model

Ronan Depoortère, Mariusz Papp, Piotr Gruca [...]

Journal of Psychopharmacology

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Research article

First published 2024-7

The 5-HT1A receptor biased agonists,NLX-204 and NLX-101,like ketamine,elicit rapid-acting antidepressant activity in the rat chronic mild stress model via cortical mechanisms

Mariusz Papp, Piotr Gruca, Ewa Litwa [...]

Journal of Psychopharmacology

Free access

Research article

First published 2017-8

A Systematic Approach to Identify Biased Agonists of the Apelin Receptor through High-Throughput Screening

Danielle McAnally, Khandaker Siddiquee, Haleli Sharir [...]

Journal of Biomolecular Screening

Open access

Research article

First published 2016

Characterization of methadone as a β-arrestin-biased μ-opioid receptor agonist

Seira Doi, Tomohisa Mori, Naoki Uzawa [...]

Molecular Pain

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Research article

First published 2017-6

Effects of acute and repeated treatment with the biased mu opioid receptor agonist TRV130 (oliceridine) on measures of antinociception,gastrointestinal function,and abuse liability in rodents

Ahmad A Altarifi, Bethany David, Karan H Muchhala [...]

Journal of Psychopharmacology

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Other

First published 2017-12

Homology Modeling of Ffa2 Identifies Novel Agonists that Potentiate Insulin Secretion

Stephanie R Villa, Rama K Mishra, Joseph L Zapater [...]

Journal of Investigative Medicine

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Review article

First published 2025-8

Biased Agonism in Incretin-based Therapies

Krishna G. Seshadri

International Journal of Clinical Metabolism and Diabetes

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Research article

First published 2025-06

The Combination of TLR4 and TLR9 Agonists with Self-Amplifying RNA Lipid Nanoparticles Leads to a More Powerful Immune Response Against SARS-CoV-2

Reza Keikha, Ebrahim Balali, Ramona Khadivi [...]

Viral Immunology

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Research article

First published 2009-08

Pharmacological Characterization of Receptor Redistribution and β-Arrestin Recruitment Assays for the Cannabinoid Receptor 1

Miranda M.C. van der Lee, Marion Blomenröhr, Antoon A. van der Doelen [...]

Journal of Biomolecular Screening

Free access

Research article

First published 2008-12

Duplexed Label-Free G Protein—Coupled Receptor Assays for High-Throughput Screening

Elizabeth Tran, Ye Fang

Journal of Biomolecular Screening

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