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Research article

First published 2015-6

Detection and Quantification of Allosteric Modulation of Endogenous M 4 Muscarinic Acetylcholine Receptor Using Impedance-Based Label-Free Technology in a Neuronal Cell Line

Amy N. Y. Chen, Daniel T. Malone, Kavita Pabreja [...]

Journal of Biomolecular Screening

Free access

Research article

First published 2014-10

Identification of Selective Agonists and Positive Allosteric Modulators for µ- and δ-Opioid Receptors from a Single High-Throughput Screen

Neil T. Burford, Tom Wehrman, Daniel Bassoni [...]

Journal of Biomolecular Screening

Free access

Research article

First published 2014-7

A Duplexed High-Throughput Screen to Identify Allosteric Modulators of the Glucagon-Like Peptide 1 and Glucagon Receptors

Lindsey C. Morris, Emily L. Days, Maxine Turney [...]

Journal of Biomolecular Screening

Free access

Research article

First published 2016-12

Identification of Positive Allosteric Modulators of Glycine Receptors from a High-Throughput Screen Using a Fluorescent Membrane Potential Assay

Clara Stead, Adam Brown, Cathryn Adams [...]

Journal of Biomolecular Screening

Retricted access

Research article

First published 2017-4

First in human trial of a type I positive allosteric modulator of alpha7-nicotinic acetylcholine receptors: Pharmacokinetics,safety,and evidence for neurocognitive effect of AVL-3288

Kelvin W Gee, Ann Olincy, Richard Kanner [...]

Journal of Psychopharmacology

Retricted access

Research article

First published 2020-1

Pharmacological characterisation of MDI-222,a novel AMPA receptor positive allosteric modulator with an improved safety profile

Simon E Ward, Mark H Harries, Laura Aldegheri [...]

Journal of Psychopharmacology

Retricted access

Review article

First published 2016-01

Allosteric Modulators of the CB 1 Cannabinoid Receptor: A Structural Update Review

Paula Morales, Pilar Goya, Nadine Jagerovic [...]

Cannabis & Cannabinoid Research

Free access

Research article

First published 2014-3

Determining the Relative Efficacy of Positive Allosteric Modulators of the GABA A Receptor

Philippe Ghisdal, Nadine Noel, Nathalie Pacico [...]

Journal of Biomolecular Screening

Open access

Research article

First published 2018-12

Exploring 6-Azaindole and 7-Azaindole Rings for Developing Cannabinoid Receptor 1 Allosteric Modulators

Sri Sujana Immadi, Rachel Dopart, Zhixing Wu [...]

Cannabis & Cannabinoid Research

Retricted access

Research article

First published 2014-5

Limited central side effects of a β-subunit subtype-selective GABA A receptor allosteric modulator

Ryan F Yoshimura, Minhtam B Tran, Derk J Hogenkamp [...]

Journal of Psychopharmacology

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