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Research article

First published 2020-3

Development of a High-Throughput Screening-Compatible Assay for Discovery of GPR3 Inverse Agonists Using a cAMP Biosensor

Kumiko Ayukawa, Chie Suzuki, Hiroyuki Ogasawara [...]

Journal of Biomolecular Screening

Open access

Brief report

First published 2008-1

The Effect of Deletion of the Orphan G – Protein Coupled Receptor (GPCR) Gene MrgE on Pain-Like Behaviours in Mice

Peter J Cox, Tom Pitcher, Steven A Trim [...]

Molecular Pain

Free access

Research article

First published 2009-08

Identification of Surrogate Agonists and Antagonists for Orphan G-Protein-Coupled Receptor GPR139

Liaoyuan A. Hu, Pauline M. Tang, Nima K. Eslahi [...]

Journal of Biomolecular Screening

Free access

Research article

First published 2013-6

Screening β-Arrestin Recruitment for the Identification of Natural Ligands for Orphan G-Protein–Coupled Receptors

Craig Southern, Jennifer M. Cook, Zaynab Neetoo-Isseljee [...]

Journal of Biomolecular Screening

Retricted access

Research article

First published 1999-03

Functional Genomics and the Discovery of New Drug Targets

Olivier Civelli, Hans-Peter Nothacker

Diabetes Technology & Therapeutics

Retricted access

Review article

First published 2003-04

G Protein-Coupled Receptors in Drug Discovery

Ponnal Nambi, Nambi Aiyar

ASSAY and Drug Development Technologies

Retricted access

Research article

First published 2007-06

Emerging Concepts of Guanine Nucleotide-Binding Protein-Coupled Receptor (GPCR) Function and Implications for High Throughput Screening

Richard M. Eglen, Roger Bosse, Terry Reisine

ASSAY and Drug Development Technologies

Retricted access

Research article

First published 2008-06

A 1,536-Well [ 35 S]GTP γ S Scintillation Proximity Binding Assay for Ultra-High-Throughput Screening of an Orphan G α i-Coupled GPCR

Eric N. Johnson, Xiaoqing Shi, Jason Cassaday [...]

ASSAY and Drug Development Technologies

Free access

Research article

First published 2007-03

Using Ligand-Induced Conformational Change to Screen for Compounds Targeting G-Protein-Coupled Receptors

Brian F. O'Dowd, Mohammad Alijaniaram, Xiaodong Ji [...]

Journal of Biomolecular Screening

Free access

Other

First published 2004-4

Multiplex GPCR Assay in Reverse Transfection Cell Microarrays

Yuji M. Mishina, Christopher J. Wilson, Linda Bruett [...]

Journal of Biomolecular Screening

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