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Research article

First published 2021-7

A Quantitative Bioassay to Determine the Inhibitory Potency of NGF–TrkA Antagonists

Francesca Malerba, Bruno Bruni Ercole, Rita Florio [...]

Journal of Biomolecular Screening

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Research article

First published 2003-01

Fluorescence Polarization Competition Assay: The Range of Resolvable Inhibitor Potency Is Limited by the Affinity of the Fluorescent Ligand

Xinyi Huang

Journal of Biomolecular Screening

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Research article

First published 2013-2

Identification of Potent VHZ Phosphatase Inhibitors with Structure-Based Virtual Screening

Hwangseo Park, So Ya Park, Jung Jin Oh [...]

Journal of Biomolecular Screening

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Research article

First published 2017-2

AKR1C3 Inhibitory Potency of Naturally-occurring Amaryllidaceae Alkaloids of Different Structural Types

Daniela Hulcová, Kateřina Breiterová, Lucie Zemanová [...]

Natural Product Communications

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Research article

First published 2006-04

Screening for Caspase-3 Inhibitors: A New Class of Potent Small-Molecule Inhibitors of Caspase-3

Ilya Okun, Sergei Malarchuk, Elena Dubrovskaya [...]

Journal of Biomolecular Screening

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Research article

First published 2010-1

Novel Potent Inhibitors of Deoxycytidine Kinase Identified and Compared by Multiple Assays

Xuan-Chuan Yu, Maricar Miranda, Ziye Liu [...]

Journal of Biomolecular Screening

Retricted access

Research article

First published 2009

Inhibitory Potency of Choline Esterase Inhibitors on Acetylcholine Release and Choline Esterase Activity in Fresh Specimens of Human and Rat Neocortex

Rolf Jackisch, Stefan Förster, Miriam Kammerer [...]

Journal of Alzheimer’s Disease

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Research article

First published 1995-10

Potent and Orally Bioavailable HIV-1 Proteinase Inhibitors Containing the 2-aminobenzylstatine Moiety

A. Billich, D. Scholz, B. Charpiot [...]

Antiviral Chemistry and Chemotherapy

Open access

Research article

First published 2016-2-22

AZD3293: A Novel,Orally Active BACE1 Inhibitor with High Potency and Permeability and Markedly Slow Off-Rate Kinetics

Susanna Eketjäll, Juliette Janson, Karin Kaspersson [...]

Journal of Alzheimer’s Disease

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Research article

First published 2007-12

A FLIPR-Based Assay to Assess Potency and Selectivity of Inhibitors of the TEC Family Kinases Btk and Itk

John Douhan, Joy S. Miyashiro, Xiaochuan Zhou [...]

ASSAY and Drug Development Technologies

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