Abstract
An efficient rapid method for the synthesis of new triazole derivatives derived from methyl 3-oxocholanate under microwave irradiation has been developed. These new compounds were characterised by 1H NMR, IR, ESI-MS spectra and elemental analyses. Some of these triazoles were tested for antibacterial activity against Staphylococcus aureus, Candida albicans and Escherichia coli.
References
1.
Amir M.
,
Kumar H.
, and
Javed S.A.
, Eur. J. Med. Chem. , 2008 , 43 , 2056 .
2.
Palaska E.
,
Sahin G.
,
Kelicen P.
,
Durlu N.T.
, and
Altinok G.
, IL Farmaco , 2002 , 57 , 101 .
3.
Tehranchian S.
,
Akbarzadeh T.
,
Fazeli M.R.
,
Jamalifar H.
, and
Shafiee A.
, Bioorg. Med. Chem. Lett. , 2005 , 15 , 1023 .
4.
Sztanke K.
,
Tuzimski T.
,
Rzymowska J.
,
Pasternak K.
, and
Kandefer-Szersze M.
, Eur. J. Med. Chem. , 2008 , 43 , 404 .
5.
Kuş C.
,
Kılcıgil G.A.
,
özbey S.
,
Kaynak F.B.
,
Kaya M.
,
Çban T.
, and
Eke B.C.
, Bioorg. Med. Chem. , 2008 , 16 , 4294 .
6.
Holla B.S.
,
Poorjary N.K.
,
Rao S.B.
, and
Shivananda M.K.
, Eur. J. Med. Chem. , 2002 , 37 , 511 .
7.
Bhat A.R.
,
Bhat G.V.
, and
Shenoy G.G.
, J. Pharm. Pharmacol. , 2001 , 53 , 267 .
8.
Demirbas N.
,
Ugurluoglu R.
, and
Demirbas A.
, Bioorg. Med. Chem. , 2002 , 10 , 3717 .
9.
Kahaveci B.
,
Bekircan O.
,
Serdar M.
, and
Ikizler A.A.
, Indian J. Chem. , Sect B., 2003 , 42B , 1527 .
10.
Demirbaş N.
,
Karaoğrlu S.A.
,
Demirbas A.
, and
Sancak K.
, Eur. J. Med. Chem. , 2004 , 39 , 793 .
11.
Demirbaş N.
, and
Uğrurluoğrlu R.
, Turk. J. Chem. , 2004 , 28 , 559 .
12.
Demirbaş N.
, and
Uğrurluoğrlu R.
, Turk. J. Chem. , 2004 , 28 , 679 .
13.
Demirbaş N.
,
Demirbas A.
, and
Karaoğrlu S.A.
, Russ. J. Bioorg. Chem. , 2005 , 31 , 430 .
14.
Virtanen E.
, and
Kolehmainen E.
, Eur. J. Org. Chem. , 2004 , 3385 .
15.
Tamminen J.
, and
Kolehmainen E.
, Molecules , 2001 , 6 , 21 .
16.
Camoutsis C.
, J. Heterocycl. Chem. , 1996 , 33 , 539 .
17.
Davidson L.
, and
Hayes W.
, Curr. Org. Chem. , 2002 , 6 , 265 .
18.
Geng L.J.
,
Feng G.L.
, and
Yu J.G.
, J. Chem. Res. , 2010 , 6 , 333 .
19.
Feng S.U.
,
Jiang S.L.
,
Zhang Z.Y.
, and
Yu X.C.
, J. Chem. Res. , 2010 , 7 , 392 .
20.
Rao M.L.N.
,
Awasthi D.K.
, and
Banerjee D.
, Tetrahedron Lett. , 2007 , 48 , 431 .
21.
Polshettiwar V.
, and
Varma R.S.
, Acc. Chem. Res. , 2008 , 41 , 629 .
22.
Zhao Z.G.
,
Liu X.L.
, and
Zhou C.E.
, Chin. Chem. Lett. , 2007 , 18 , 1067 .
23.
Colacino E.
,
Lamaty F.
,
Martinez J.
, and
Parrot I.
, Tetrahedron Lett. , 2007 , 48 , 5317 .
24.
Zhou C.E.
,
Zhao Z.G.
, and
Tang X.L.
, Chin. J. Org. Chem. , 2007 , 4 , 513 . (in Chinese).
25.
Fieser L.F.
, and
Rajagopalan S.
, J. Am. Chem. Soc. , 1950 , 72 , 5530
26.
Cui J.G.
,
Huang L.L.
,
Huang Y.M.
, and
Fan J.C.
, Chin. J. Org. Chem. , 2009 , 6 , 971 . (in Chinese).
27.
Fieser L.F.
, and
Ettorce R.
, J. Am. Chem. Soc. , 1953 , 75 , 1700 .
28.
Khan M.
,
Hameed S.
,
Yasin K.A.
,
Akhtar T.
, and
Khan K.M.
, Monatsh. Chem. , 2010 , 141 , 479 .
29.
Eweiss N.F.
,
Bahajaj A.A.
, and
Elsherbini E.A.
, J. Heterocycl. Chem. , 1986 , 23 , 1451 .
30.
Jag M.
, Indian J. Chem. , Sect B., 1990 , 29B , 88 .
