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Research article

First published 2020-3

Development of a High-Throughput Screening-Compatible Assay for Discovery of GPR3 Inverse Agonists Using a cAMP Biosensor

Kumiko Ayukawa, Chie Suzuki, Hiroyuki Ogasawara [...]

Journal of Biomolecular Screening

Retricted access

Research article

First published 2025-7

Interactions of alcohol and the benzodiazepine inverse agonist in healthy male volunteers

Nirmal Singh, Ismene Petrakis, Brian Pittman [...]

Journal of Psychopharmacology

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Research article

First published 1993-1

Pre-natal benzodiazepine exposure. III. Lorazepam exposure is associated with a shift toward inverse agonist efficacy

John J. Byrnes, Lawrence G. Miller

Journal of Psychopharmacology

Open access

Research article

First published 2011-8

Specific targeting of the GABA-A receptor α5 subtype by a selective inverse agonist restores cognitive deficits in Down syndrome mice

J Braudeau, B Delatour, A Duchon [...]

Journal of Psychopharmacology

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Research article

First published 2012-2

The effects of a novel histamine-3 receptor inverse agonist on essential tremor in comparison to stable levels of alcohol

RWM Zoethout, R Iannone, BR Bloem [...]

Journal of Psychopharmacology

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Research article

First published 2010-08

Strategy for the Identification of GPR23/LPA 4 Receptor Agonists and Inverse Agonists

Soo Hang Wong, Rommel Mallari, Melissa Graham [...]

ASSAY and Drug Development Technologies

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Research article

First published 1996-7

Benzodiazepine receptor agonists and inverse agonists yield concordant rather than opposing effects on startle responses

G. Berntson, M. Sarter, S. Ruland [...]

Journal of Psychopharmacology

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Research article

First published 2018-06

Cholesterol Unbound RORγt Protein Enables a Sensitive Inverse Agonist Screening

Ryokichi Koyama, Yasunori Fukuda, Yusuke Kamada [...]

ASSAY and Drug Development Technologies

Open access

Research article

First published 2016-12

CB 1 Allosteric Modulator Org27569 Is an Antagonist/Inverse Agonist of ERK1/2 Signaling

Thomas F. Gamage, Johnathon C. Anderson, Mary E. Abood

Cannabis & Cannabinoid Research

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Research article

First published 2025

Cannabinoid 1 receptor occupancy and neurovascular responses induced by agonist,antagonist/inverse-agonist,and potential modulator in non-human primate brains: PET/fMRI study

Chi-Hyeon Yoo, Yulong Xu, Frederick A Bagdasarian [...]

Journal of Cerebral Blood Flow & Metabolism

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