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Research article

First published 2003-10

Development of Displacement Binding and GTPγS Scintillation Proximity Assays for the Identification of Antagonists of the μ-Opioid Receptor

George Rodgers, Cassandra Hubert, Jamie McKinzie [...]

ASSAY and Drug Development Technologies

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Research article

First published 2003-04

A Fully Automated [ 35 S]GTPγS Scintillation Proximity Assay for the High-Throughput Screening of G i -Linked G Protein-Coupled Receptors

Marc Ferrer, Garrett D. Kolodin, Paul Zuck [...]

ASSAY and Drug Development Technologies

Free access

Research article

First published 2007-04

Evaluation of Cellular Dielectric Spectroscopy,a Whole-Cell,Label-Free Technology for Drug Discovery on G i -Coupled GPCRs

Matthew F. Peters, Katharine S. Knappenberger, Deidre Wilkins [...]

Journal of Biomolecular Screening

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Research article

First published 2005-05

Trazodone and its active metabolite m-chlorophenylpiperazine as partial agonists at 5-HT1A receptors assessed by [35S]GTPγS binding

Yuji Odagaki, Ryoichi Toyoshima, Toshio Yamauchi

Journal of Psychopharmacology

Free access

Research article

First published 2014-3

No Differences Observed among Multiple Clinical S1P 1 Receptor Agonists (Functional Antagonists) in S1P 1 Receptor Down-regulation and Degradation

Susan Lukas, Lori Patnaude, Sokol Haxhinasto [...]

Journal of Biomolecular Screening

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Other

First published 2010-05

The cannabinoid CB1 receptor is involved in the anxiolytic,sedative and amnesic actions of benzodiazepines

María S García-Gutiérrez, Jorge Manzanares

Journal of Psychopharmacology

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Research article

First published 2010-10

A Homogeneous Method to Measure Nucleotide Exchange by α-Subunits of Heterotrimeric G-Proteins Using Fluorescence Polarization

Robin E. Muller, Klara R. Klein, Stephanie Q. Hutsell [...]

ASSAY and Drug Development Technologies

Free access

Research article

First published 2011-8

Understanding the Effect of Different Assay Formats on Agonist Parameters: A Study Using the µ-Opioid Receptor

Sarah A. Nickolls, Alison Waterfield, Rachael E. Williams [...]

Journal of Biomolecular Screening

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Research article

First published 2009-02

High-Throughput Screening for Small-Molecule Inhibitors of LARG-Stimulated RhoA Nucleotide Binding via a Novel Fluorescence Polarization Assay

Chris R. Evelyn, Timothy Ferng, Rafael J. Rojas [...]

Journal of Biomolecular Screening

Free access

Research article

First published 1998-03

Development of Flashplate™ Technology to Measure [35S]GTPyS Binding to Chinese Hamster Ovary Cell Membranes Expressing the Cloned Human 5-HTIB Receptor

J. Watson, J. V. Selkirk, A. M. Brown

Journal of Biomolecular Screening

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