Abstract
Some new derivatives of 2-arylthieno[2,3-d]pyrimidin-4(3H)-ones have been prepared through a condensation reaction of 2-amino-4,5-dimethylthiophene-3-carboxamide with aroyl halides in boiling pyridine followed by cyclisation with 10% NaOH.
Keywords
References
1.
Pathak U.S.
,
Singh S.
, and
Padh J.
, Indian J. Chem., Sect B , 1991 , 30B , 618 .
2.
Rathod I.S.
,
Pillai A.S.
, and
Shirsath V.S.
, Indian J. Heterocycl. Chem. , 2000 , 10 , 93 .
3.
Kharizomenova I.A.
,
Grinev A.N.
,
Samsonova N.V.
,
Panisheva E.K.
,
Kaplina N.V.
,
Nikolaeva I.S.
,
Pushkina T.V.
, and
Pershin G.N.
, Khim.-Farm. Zh. , 1981 , 15 , 40 .
4.
Showa D.K.K.
, Jpn. Kokai. Tokkyo. Koho. 81,53,681, 1981, Chem. Abstr. , 1981 , 95 , 115592y .
5.
Perrissin M.
,
Favre M.
,
Luu-Duc C.
,
Bakri-Logeais F.
,
Huguet F.
, and
Narcisse G.
, Eur. J. Med. Chem - Chim. Ther. , 1984 , 19 , 420 .
6.
El-Ansary A.K.
, and
Omar A.H.
, Bull. Fac. Pharm. , 2001 , 39 , 17 .
7.
Pathak U.S.
,
Gandhi N.V.
,
Singh S.
,
Warde R.P.
, and
Jain K.S.
, Indian J. Chem., Sect B , 1992 , 31B , 223 .
8.
Donkor I.O.
,
Li H.
, and
Queener Sh.F.
, Eur. J. Med. Chem. , 2003 , 38 , 605 .
9.
Matsuda T.
,
Yamazaki K.
,
Ide H.
,
Noda K.
, and
Yamagata K.
, Japan. Kokai. 74,11,895, 1974, Chem. Abstr. , 1974 , 80 , 108567f .
10.
Hiroyashi T.
,
Sato H.
,
Inaba S.
, and
Yamamoto H.
, Ger. Offen. 2,323,149, 1973, Chem. Abstr. , 1974 , 80 , 70825y .
11.
Wiesenfeldt M.
,
Etzbach K.H.
,
Hofmeister P.
,
Kuenast C.
, and
Westphalen K.O.
, Eur. Pat. Appl. EP. 447,891, Chem. Abstr. , 1991 , 115 , 256224y .
12.
Shishoo C.J.
,
Devani M.B.
,
Pathak U.S.
,
Ananthan S.
,
Bhadti V.S.
,
Ullas G.V.
,
Jain K.S.
,
Rathod I.S.
,
Talati D.S.
, and
Doshi N.H.
, J. Heterocycl. Chem. , 1984 , 21 , 375 .
13.
Csuros Z.
,
Soos R.
,
Palinkas J.
, and
Bitter I.
, Acta. Chim (Budapest). , 1971 , 68 , 397 .
14.
Sauter F.
, Monatsh. Chem. , 1970 , 101 , 535 .
15.
Link H.
, Helv. Chim. Acta. , 1990 , 73 , 797 .
16.
Gakhar H.K.
, and
Gill J.K.
, Indian J. Chem., Sect B , 1985 , 24B , 432 .
17.
Rahimizadeh M.
,
Davoodnia A.
,
Heravi M.M.
, and
Bakavoli M.
, Phosphorus, Sulfur and Silicon. , 2002 , 177 , 2923 .
18.
Bakavoli M.
,
Davoodnia A.
,
Rahimizadeh M.
,
Heravi M.M.
, and
Ghassemzadeh M.
, J. Chem. Res., (S) , 2002 , 1 , 178 .
19.
Bakavoli M.
,
Davoodnia A.
,
Rahimizadeh M.
, and
Heravi M.M.
, Phosphorus, Sulfur Silicon , 2002 , 177 , 2303 .
20.
Roshani M.
,
Davoodnia A.
,
Hedayat M. Sh.
, and
Bakavoli M.
, Phosphorus, Sulfur Silicon , 2004 , 179 , 1153 .
21.
Davoodnia A.
,
Zhiani R.
,
Roshani M.
,
Bakavoli M.
, and
Bashash M.
Phosphorus, Sulfur Silicon , 2007 , 182 , 1219 .
22.
Davoodnia A.
,
Momen-Heravi M.
,
Golshani E.
,
Bakavoli M.
, and
Dehabadi L.
, J. Chem. Res. , 2007 , 257 .
23.
Davoodnia A.
,
Behmadi H.
,
Zare-Bidaki A.
,
Bakavoli M.
, and
Tavakoli-Hoseini N.
, Chin. Chem. Lett. , 2007 , 18 , 1163 .
24.
Davoodnia A.
,
Bakavoli M.
,
Barakouhi Gh.
, and
Tavakoli-Hoseini N.
, Chin. Chem. Lett. , 2007 , 18 , 1483 .
25.
Sauter F.
, and
Deinhammer W.
, Monatsh. Chem. , 1973 , 104 , 1586 .
